Dofetilide effect on human atrial action potential under normal and atrial fibrillation conditions. In silico study

Catalina Tobón, S. Pérez, J. P. Ugarte, J. Saiz

Producción científica: Capítulo del libro/informe/acta de congresoContribución a la conferenciarevisión exhaustiva

2 Citas (Scopus)

Resumen

Atrial fibrillation is the most common sustained cardiac arrhythmia. Dofetilide is an antiarrhythmic drug for the treatment of chronic AF that specifically blocks the rapid component of the delayed rectifier potassium current IKr. Dofetilide prolongs the action potential duration and QT interval in a concentration-dependent fashion, therefore, the risk of QT prolongation is dose related. It is important to study the electrophysiological effects of dofetilide at different concentrations in human atrial cells. For this, we simulated the effects of dofetilide on human atrial cell and studied its effect on atrial action potential under normal conditions and during cAF. We developed a model of dofetilide effects on IKrand IKACh. Our results show that dofetilide blocks both currents in a fraction greater as the concentration increases, which results in an action potential duration lengthening. To our knowledge, this is the first work that has developed mathematical models of dofetilide effects on IKrand IKAChcurrents to study its effect on human atrial action potential.

Idioma originalInglés
Título de la publicación alojada7th Latin American Congress on Biomedical Engineering, CLAIB 2016
EditoresJohn Bustamante, Daniel A. Sierra, Isnardo Torres
EditorialSpringer Verlag
Páginas38-41
Número de páginas4
ISBN (versión impresa)9789811040856
DOI
EstadoPublicada - 2017
Publicado de forma externa
Evento7th Latin American Congress on Biomedical Engineering, CLAIB 2016 - Bucaramanga, Santander, Colombia
Duración: 26 oct. 201628 oct. 2016

Serie de la publicación

NombreIFMBE Proceedings
Volumen60
ISSN (versión impresa)1680-0737

Conferencia

Conferencia7th Latin American Congress on Biomedical Engineering, CLAIB 2016
País/TerritorioColombia
CiudadBucaramanga, Santander
Período26/10/1628/10/16

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